CBP bromodomain inhibitor ( —— )

产品货号. M13447 CAS No. 2161356-61-0

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

CBP bromodomain inhibitor
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

a potent, selective CBP bromodomain inhibitor with IC50 of 69 nM, displays exquisite selectivity over BRD4(1) (IC50=18 uM) and the broader bromodomain family.
产品描述

a potent, selective CBP bromodomain inhibitor with IC50 of 69 nM, displays exquisite selectivity over BRD4(1) (IC50=18 uM) and the broader bromodomain family.
同义词

——
通路

Chromatin/Epigenetic
靶点

Bromodomain
受体

Bromodomain
研究领域

——
适应症

——

CAS Number

2161356-61-0
分子量

426.49
分子式

C22H20F2N4OS
纯度

>98% (HPLC)
溶解度

——
SMILES

——
化学全称

5-(7-(difluoromethyl)-6-(1-methyl-1H-pyrazol-4-yl)-3,4-dihydroquinolin-1(2H)-yl)-3-methylbenzo[d]thiazol-2(3H)-one

1. Bronner SM, et al. J Med Chem. 2017 Dec 28;60(24):10151-10171.

计算器

产品手册

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